0. Twist1 run — DONE

0. Twist1 run — DONE

Status: the databases were downloaded and the Twist1 run completed. Full network: 17,191 genes / 1,891,745 directed edges (IID mouse PPI + TRRUST v2 regulatory edges). Driver Twist1; 168/182 RNA-seq response genes in-network (14 absent from the interactome). Dense NetPert (nt=16, r=0.5) on a 1,200-gene Twist1-centered subnetwork (228,199 edges); conservation identity max rel. deviation 1.99e-15. Betweenness run on the full 17k-gene network. 1,182 genes mapped to Drug Repurposing Hub compounds. Full outputs: geneRankings_real.tsv · summary_real.json · figure gallery. The simulation sections below are unchanged and test algorithm behaviour only; biological claims rest on this section.
#GeneNetPert weightBC-sub rankRepurposing compounds (sample)
1Pdgfra2.13e-023AC-710, BMS-536924, CP-673451, DCC-2618
2Htt1.80e-021—
3Tp531.76e-024—
4Ctnnb11.53e-026CCT-031374, ICG-001, PNU-74654, cardionogen-1
5Cdh11.51e-025—
6Zranb11.43e-022—
7Vim1.37e-027—
8Ppia1.36e-0227L-proline, TMN-355, cyclosporin-A
9Stat31.28e-0210APcK-110, STAT3-inhibitor-VI, WP1066, acitretin
10Clu1.28e-0220—
11Stub11.26e-0225—
12Nfkb11.25e-0217SP-100030, andrographolide, arglabin, aspirin
13Ep3001.15e-0214C646, I-CBP-112, SGC-CBP30, curcumin
14Sox21.14e-028—
15Col2a11.08e-029—
16Rela1.08e-0219BAY-11-7082, NFKB-activation-inhibitor-II, acetylcysteine, bortezomib
17Kif231.07e-0221—
18Hif1a1.04e-02402-methoxyestradiol, 3, 3'-diindolylmethane, BAY-87-2243
19Hdac61.02e-0215ACY-1215, JNJ-26481585, PCI-24781, PCI-34051
20H4c11.02e-0212—

Top-20 NetPert intermediates from the IID+TRRUST Twist1 network (all type I). Assay check (honest null): 18 genes have both a ranking and a dissemination readout; Spearman(NetPert, dissemination %) = +0.31, p=0.21; BC = −0.10. All 18 are response genes while NetPert prioritises intermediates, so the test is underpowered by construction.

 figure
Top-20 NetPert intermediates, weights.
 figure
Response coverage: 168/182 DE genes in-network; network sizes.
 figure
NetPert vs full-network betweenness (Spearman rho=0.59, n=1200).
 figure
Hub-bias check: out-degree vs NetPert (rho=0.51).
 figure
dissemination % at 1 µM for the 18 assayed genes.
 figure
NetPert vs dissemination (n=18, rho=+0.31, p=0.21, not significant).

Highlights above. The full gallery holds all 100 grouped visuals: rankings (11) · network (11) · assays (13) · gene spotlights top-40 (40) · drugs (12) · method comparison (11) · overview (2).

0.2 Full ranking: all 1,200 genes (embedded)

Show all 1,200 ranked genes
NetPert rankGeneTypeNetPert weightBC-sub rankBC-full weightOut-degreeDrugs
1PdgfraI2.126e-0236.170e+00373AC-710,BMS-536924,CP-673451,DCC-2618,ENMD-2076,PD-173074,PP-121,TAK-593,cediranib,crenolanib
2HttI1.800e-0217.683e+001523
3Tp53I1.757e-0245.596e+002321
4Ctnnb1I1.535e-0264.285e+001236CCT-031374,ICG-001,PNU-74654,cardionogen-1,iCRT-14,urea
5Cdh1I1.513e-0254.708e+00933
6Zranb1I1.433e-0226.641e+003868
7VimI1.374e-0274.089e+00863
8PpiaI1.365e-02271.780e+00883L-proline,TMN-355,cyclosporin-A
9Stat3I1.277e-02103.175e+00618APcK-110,STAT3-inhibitor-VI,WP1066,acitretin,alantolactone,atiprimod,bardoxolone-methyl,cryptotanshinone,meisoindigo,napabucasin
10CluI1.277e-02202.243e+00310
11Stub1I1.260e-02251.905e+00691
12Nfkb1I1.251e-02172.274e+00683SP-100030,andrographolide,arglabin,aspirin,pranlukast,triflusal
13Ep300I1.147e-02142.422e+001371C646,I-CBP-112,SGC-CBP30,curcumin,epigallocatechin-gallate-(-)
14Sox2I1.144e-0283.838e+001386
15Col2a1I1.085e-0293.654e+0070
16RelaI1.076e-02192.269e+00679BAY-11-7082,NFKB-activation-inhibitor-II,acetylcysteine,bortezomib,caffeic-acid-phenethyl-ester,parthenolide-(alternate-stereo),pyrrolidine-dithiocarbamate,triptolide
17Kif23I1.071e-02212.136e+00965
18Hif1aI1.038e-02401.319e+004642-methoxyestradiol,3,3'-diindolylmethane,BAY-87-2243,FG-2216,ML228,YC-1,acriflavine,acriflavinium,bakuchiol,melphalan-n-oxide
19Hdac6I1.021e-02152.157e+00861ACY-1215,JNJ-26481585,PCI-24781,PCI-34051,SB-939,TCS-HDAC6-20b,belinostat,bufexamac,dacinostat,droxinostat
20H4c1I1.018e-02122.610e+001833
21PdgfrbI1.014e-02441.346e+00304AC-710,BMS-536924,CP-673451,GTP-14564,KG-5,KI-20227,MK-2461,ON123300,PD-166285,PD-173074
22Stau1I9.532e-03132.507e+001463
23Hdac1I9.460e-03541.123e+0011164SC-202,ACY-1215,AR-42,JNJ-26481585,Merck60,NSC-3852,PCI-24781,PCI-34051,RG2833,SB-939
24IkbkbI9.440e-03501.196e+00302AZD3264,BMS-345541,IKK-16,IKK-2-inhibitor,IKK-2-inhibitor-V,PF-573228,TPCA-1,acetylcysteine,arsenic-trioxide,aspirin
25TnfI9.163e-03181.887e+00387CPI-1189,JTE-607,SB-203580,VX-702,amrinone,andrographolide,baicalein,bergenin,ephedrine-(racemic),epinephrine
26Eif2b5I8.659e-03351.464e+00207
27Cul4aI8.578e-03261.943e+00790
28Hdac2I8.532e-03678.006e-01878ACY-1215,CUDC-907,JNJ-26481585,MC1568,Merck60,PCI-24781,SB-939,TC-H-106,UF-010,aminophylline
29Esr1I8.392e-03113.191e+00230517-hydroxyprogesterone-caproate,AZD9496,GDC-0810,PPT,SNG-1153,Y-134,ZK-164015,afimoxifene,allylestrenol,bazedoxifene
30Ppp2caI8.317e-03481.287e+00516vitamin-E
31Mcm7I8.287e-03431.280e+00527
32ZyxR8.201e-03757.899e-01338
33Tcf4I8.169e-03985.949e-01368PNU-74654,iCRT-14
34Tcf3I8.138e-03242.082e+00316
35FosI7.915e-03311.674e+00449ephedrine-(racemic)
36Ilf3I7.419e-03461.191e+001147
37Obsl1I7.094e-03659.389e-01831
38Epha3I7.031e-03281.668e+00112vandetanib
39Trp53I7.011e-03361.401e+00166APR-246,PhiKan-083,VLX600,aspirin,carbendazim,idasanutlin,nutlin-3,pifithrin-alpha,pifithrin-cyclic,pifithrin-mu
40Hk2I6.903e-03638.793e-011593-bromopyruvate
41Bcl6I6.895e-03222.102e+00255
42BtrcI6.878e-03907.418e-01750GS-143
43Skp2I6.630e-031304.529e-01296
44Fkbp4I6.554e-03381.441e+00284
45Atp2a2I6.515e-03301.660e+00403gallopamil
46Tubg1I6.397e-03511.075e+00381vinblastine
47Ythdf1I6.346e-03708.135e-01423
48Rbbp7I6.065e-03867.050e-01501
49Ppp1ccI5.717e-03877.060e-01731
50VegfaI5.578e-03738.349e-0180pidolic-acid,trometamol,vandetanib
51Fbxo45I5.420e-03916.649e-0196
52Fgfr2I5.402e-03647.282e-01233AEE788,AZD4547,CH-5183284,LY2874455,MK-2461,NVP-BGJ398,PD-173074,RG1530,dovitinib,erdafitinib
53Fosl1I5.359e-03232.091e+0096
54Dnajb6I5.274e-03371.504e+00444
55Wdr5I5.265e-03321.426e+001047OICR-9429,WDR5-0103
56Trim28I5.249e-03341.479e+001310
57BcorI5.242e-03957.094e-01300
58Ubr5I5.234e-03559.465e-01554
59Usp4I5.164e-031214.987e-01273
60Cdkn1aI5.163e-031742.882e-01368GGTI-298
61Vdac2I5.042e-03838.080e-01503erastin
62Rad23aI5.041e-031154.504e-01267
63MgaI5.013e-031374.385e-01236
64Myod1I4.998e-031643.161e-01234
65Ythdf2I4.994e-031254.464e-01454
66Yy1I4.963e-03411.269e+00469
67Dnaja2I4.927e-03748.190e-01865
68Rnf8I4.897e-031045.923e-01380
69Dhx30I4.760e-03856.907e-01545
70Brd4I4.610e-03667.994e-011482ARV-825,BI-2536,CPI-0610,CPI-203,I-BET-762,I-BET151,JQ1-(+),LY303511,OTX015,OXF-BD-02
71Brd7I4.460e-031115.612e-01611
72Cdk9I4.258e-031274.539e-01745AT-7519,BMS-387032,CDK9-IN-6,LY2857785,P276-00,PHA-793887,RGB-286638,TG-02,alvocidib,dinaciclib
73Nup155I4.152e-03291.594e+00509
74Arhgef2I4.136e-03629.331e-01278
75Xpo5I3.993e-031085.579e-01272
76Rabgap1I3.939e-03689.027e-01205
77Dnajc7I3.806e-031225.813e-01457
78Hdac3I3.796e-031882.248e-01340ACY-1215,JNJ-26481585,PCI-24781,RG2833,RGFP966,SB-939,SBHA,TC-H-106,UF-010,belinostat
79BrapI3.780e-03777.276e-0199
80CkmI3.759e-03471.300e+0071creatine,guanidinopropionic-acid
81Rps27aI3.746e-03976.723e-01724
82Nsd1I3.727e-03827.050e-01111
83Hoxa9I3.725e-031622.981e-0162
84Hspa8I3.704e-03946.521e-01210gentamycin
85Uhrf1I3.704e-031712.592e-01208
86Fgf2I3.687e-03966.784e-0161
87LbrI3.682e-031354.325e-01322
88Kat5I3.681e-031464.673e-01481coenzyme-A
89Tcf12I3.674e-031842.322e-01161
90Cul4bI3.663e-031573.422e-01684
91Ets2I3.661e-031483.731e-0189
92RalyI3.646e-031393.648e-01367
93Arrdc3I3.633e-031454.547e-01220
94Usp51I3.630e-03451.273e+0046
95Kat2bI3.616e-031692.893e-01254coenzyme-A,epigallocatechin-gallate-(-)
96Chd7I3.606e-031632.935e-01169
97Rif1I3.602e-031803.030e-01305
98G3bp2I3.584e-031343.842e-01460
99Uhrf2I3.545e-032171.509e-01197
100NfibI3.451e-031234.663e-01659
101Ddx24I3.436e-03391.333e+00588
102MaxI3.430e-031852.184e-01270
103Chd3I3.423e-03521.093e+00701
104NgefI3.359e-032051.620e-01102
105Trim67I3.150e-031403.518e-014470
106C1qbpI2.772e-03727.579e-01829hyaluronic-acid
107Psmc3I2.764e-03331.443e+00595
108Supt16hI2.684e-031363.618e-01562
109Mta2I2.626e-031533.213e-01431
110Chd4I2.571e-031065.171e-01833
111Gtpbp4I2.473e-031333.287e-01507
112Chd8I2.439e-031104.075e-01292
113Ftsj3I2.397e-031553.176e-01452
114Smarce1I2.389e-031732.398e-01318
115Gnl3lI2.317e-031563.403e-01138
116Bop1I2.286e-03896.321e-01282
117Chd1I2.238e-031961.821e-01117epirubicin
118UbtfI2.235e-031921.760e-01236
119Ehmt2I2.221e-031244.463e-01327A-366,BIX-01294,BRD4770,UNC0224,UNC0321,UNC0631,UNC0638,UNC0642,UNC0646,UNC0737
120Rrp1bI2.198e-031603.183e-01620
121Zbtb33I2.186e-032381.634e-01131
122WizI2.172e-032071.647e-01223
123Nav1I2.145e-031942.055e-01165
124Neil3I2.119e-03531.075e+0090
125Sox10I2.113e-033337.939e-02108
126Elf2I2.106e-031902.201e-01161
127Sin3bI2.104e-032391.392e-01154
128Gnl2I2.104e-031951.457e-01444
129Nsd3I2.094e-031582.630e-01121
130Kif20bI2.055e-032271.455e-01103
131Chd9I2.047e-031702.754e-0178
132Gli3I2.046e-032111.587e-01104
133Dvl1I2.038e-032371.676e-01153
134PhipI2.028e-032041.609e-01188
135Prr12I2.026e-031672.651e-0187
136TekI2.025e-032641.366e-01128ACTB-1003,altiratinib,linifanib,pexmetinib,ponatinib,regorafenib,vandetanib
137NvlI1.970e-032451.231e-01224
138Tead4I1.937e-032521.657e-0187
139Cetn1I1.933e-033771.779e-0278
140Zic3I1.926e-032331.503e-0136
141Paqr3I1.913e-031493.734e-0128
142Usp18I1.903e-032481.267e-0171
143Tbx21I1.899e-032501.210e-0132
144PostnI1.895e-031175.276e-0116
145Lin54I1.882e-033046.220e-02126
146VirmaI1.854e-03161.573e+002640
147Chmp2aI1.841e-032431.496e-01126
148Zfp62I1.810e-032769.545e-0298
149MmeR1.800e-03992.200e-01137KBG,omapatrilat,racecadotril,sacubitril,thiorphan
150Cul3I1.785e-03846.297e-012902
151Crabp1R1.675e-032699.775e-0218
152Myl6I1.459e-031543.387e-01304
153EgfrI1.451e-031005.341e-011990AEE788,AG-490,AP26113,AST-1306,AV-412,AZ5104,AZD3759,AZD8931,BIBU-1361,BIBX-1382
154UbcI1.359e-031025.757e-012436
155CftrI1.348e-033025.887e-023298CFTRinh-172,IOWH032,apigenin,bumetanide,capsaicin,dexfosfoserine,felodipine,genistein,glafenine,glyburide
156Trim25I1.277e-031074.840e-012146
157PrknI1.175e-033880.000e+003280
158Fancd2I1.117e-03766.353e-012048
159AppI1.049e-037590.000e+0026562,4-dinitrophenol,EUK-134,MRK-560,Ro-90-7501,SEN-1269,TC-E-5006,beta-amyloid-synthesis-inhibitor,curcumin,salidroside,tramiprosate
160Rpa1I1.040e-032291.400e-012924
161Trip12I1.018e-032061.432e-01239
162Usp7I1.015e-031134.147e-011469NSC-632839,P22077,P5091
163Ebna1bp2I1.005e-031861.623e-01359
164DekI9.929e-042201.320e-01277
165Rrs1I9.853e-042021.704e-01397
166Esr2I9.717e-042976.061e-02238917-hydroxyprogesterone-caproate,AC-186,C11-Acetate,PHTPP,WAY-200070,Y-134,ZK-164015,afimoxifene,bazedoxifene,bisphenol-A
167HnrnplI9.670e-04697.539e-011804
168VcpI9.661e-044580.000e+001811CB-5083,NMS-873
169Parp1I9.427e-044870.000e+0012803-amino-benzamide,4-HQN,AG-14361,BYK-204165,DR-2313,E7449,EB-47,NU-1025,PJ-34,S-111
170Pbrm1I9.230e-041981.589e-01291PFI-3
171JunI8.867e-046040.000e+001670SP-100030,T-5224,TWS-119,arsenic-trioxide,ephedrine-(racemic),irbesartan,vinblastine
172Sting1I8.725e-041055.109e-011928
173Ezh2I8.446e-04786.179e-0114843-deazaneplanocin-A,CPI-169,CPI-360,EI1,EPZ005687,EPZ011989,GSK2816126,GSK503,UNC1999,tazemetostat
174Nsd2I8.399e-042141.671e-01256
175Rpa3I8.266e-042421.277e-012723
176MaptI8.076e-041591.858e-012123docetaxel,leucomethylene-blue,paclitaxel
177Kif14I8.056e-042231.381e-011681
178Ntrk1I7.992e-041652.401e-011995GNF-5837,GW-441756,GW-5074,MK-2461,PHA-848125,amitriptyline,danusertib,entrectinib,imatinib,larotrectinib
179Rpa2I7.991e-043940.000e+002744
180St13I7.975e-042581.483e-01210
181SpenI7.495e-042549.124e-02206
182Atg16l1I7.370e-042747.973e-021997
183Zeb1I7.247e-043065.263e-02201
184Smad4I7.185e-049800.000e+00882
185CfdI7.112e-041163.933e-011417BCX-1470
186Elavl1I7.087e-041384.035e-011954
187Plekha4I7.024e-048390.000e+002796
188Top3bI6.979e-04885.375e-011426
189Fndc5I6.910e-041193.802e-011495
190Rnf4I6.910e-043283.463e-021288
191Atxn1I6.499e-044790.000e+001184
192CitI6.404e-041682.843e-011297
193PccbI6.357e-042857.136e-02165biotin
194Tgoln1I6.341e-041871.747e-011543
195AnlnI6.309e-042807.846e-021625
196SrcI6.257e-041431.888e-017421-naphthyl-PP1,3,4-methylenedioxy-beta-nitrostyrene,AZM-475271,ENMD-2076,KB-SRC-4,KX2-391,PD-166285,PD-168393,PP-121,PP-2
197Mecp2I6.249e-041323.544e-011271
198Raf1I6.238e-042121.515e-011875AZ-628,CEP-32496,GW-5074,LY3009120,ML786,PD-98059,Ro-5126766,SB-203580,U-0126,ZM-336372
199Fn1I6.230e-04924.291e-01795
200YwhazI6.215e-043930.000e+001597
201Kdm1aI6.142e-046010.000e+00920GSK-LSD-1,GSK2879552,OG-L002,ORY-1001,RN-1,tranylcypromine
202Smarca4I6.138e-048590.000e+00723PFI-3
203ActbI6.090e-041811.635e-011155cytochalasin-B
204Anp32eI6.061e-042958.351e-02132
205Sox9I5.992e-042839.625e-02134
206Erbb2I5.961e-042441.194e-01752AEE788,ARRY-334543,AST-1306,AV-412,AZD8931,BIBX-1382,BMS-536924,BMS-599626,BMS-690514,CP-724714
207Sp1I5.878e-045550.000e+00626
208Sqstm1I5.850e-041991.175e-011293
209Rbm19I5.798e-042351.169e-01242
210CebpbI5.681e-046490.000e+001382
211CcnfI5.660e-044020.000e+001945
212Hspa4I5.639e-049050.000e+00688
213Fbxw7I5.552e-043960.000e+001236
214LmnaI5.542e-041971.452e-011293
215ArI5.476e-047070.000e+0099717-hydroxyprogesterone-caproate,2-hydroxyflutamide,3,3'-diindolylmethane,APC-100,ASC-J9,AZD3514,CB-03-01,GLPG0492,GLPG0492-R-enantiomer,LXR-623
216Usp13I5.432e-042401.315e-01108spautin-1
217BbxI5.416e-042689.755e-02126
218HnrnpdI5.301e-04491.018e+001106
219RigiI5.277e-04421.068e+001595
220Zeb2I5.267e-042499.950e-02114
221Phf2I5.112e-042558.991e-0284
222Mdm2I5.060e-048860.000e+00651AMG-232,CGM097,JNJ-26481585,RG7112,RITA,SAR405838,SP-141,idasanutlin,nutlin-3,serdemetan
223Hsp90aa1I5.018e-048090.000e+001275AT13387,BIIB021,CCT018159,EC-144,NVP-AUY922,NVP-HSP990,PU-H71,SNX-5422,VER-49009,alvespimycin
224Plk1I4.949e-043084.854e-02913BI-2536,GSK461364,GW-843682X,HMN-214,LY294002,NMS-1286937,SBE-13,TAK-960,rigosertib,volasertib
225Afg2bI4.937e-045330.000e+001243
226CebpaI4.933e-041313.299e-011205
227Akt1I4.928e-043174.329e-029334,5,6,7-tetrabromobenzotriazole,A-674563,API-1,AT13148,AZD5363,BMS-536924,BMS-754807,CaMKII-IN-1,GDC-0068,GSK2110183
228Hsp90ab1I4.867e-0410400.000e+001227CCT018159,EC-144,NVP-AUY922,NVP-HSP990,SNX-5422
229NclI4.839e-042101.294e-01828
230Trib3I4.823e-042709.049e-02145
231Kctd13I4.819e-042261.230e-011490
232Ahdc1I4.817e-042461.519e-0181
233Ctbp1I4.748e-043234.069e-02793
234Smad3I4.722e-047470.000e+00511SIS3
235CanxI4.717e-042251.071e-011275
236Apex1I4.647e-047430.000e+001219lucanthone,methoxyamine
237Bmi1I4.573e-045480.000e+001171
238Calm1I4.469e-044760.000e+00900aprindine,chlorpromazine,cinchocaine,flunarizine,fluphenazine,loperamide,melatonin,nifedipine,perphenazine,pimozide
239Calm3I4.466e-048180.000e+00892
240Calm2I4.465e-049500.000e+00894
241Hspa5I4.444e-041093.782e-011559aspirin
242RhoaI4.385e-042415.566e-021182Y16
243Hectd1I4.381e-042341.117e-01948
244Chd6I4.378e-042667.997e-0279
245Fzr1I4.354e-046510.000e+001122
246Cdc42I4.321e-048760.000e+001322ML141,ZCL-278,casin
247TiparpI4.306e-044430.000e+001474
248Dyrk1aI4.282e-047960.000e+001018KH-CB19,TC-S-7004,TG-003
249Hnrnph1I4.273e-044360.000e+001413
250PrnpI4.237e-04588.056e-011117
251Ace2I4.205e-049490.000e+00998ORE1001,lisinopril,moexipril
252CrebbpI4.100e-048610.000e+00630I-CBP-112,SGC-CBP30
253Brca1I4.063e-042935.825e-021196
254Rack1I4.049e-042211.130e-01935
255Xpo7I4.042e-043323.020e-021335
256Xpo1I4.041e-045110.000e+001670KPT-185,KPT-276,elactocin,selinexor
257Yap1I4.017e-047330.000e+001042
258PrkdcI4.001e-044300.000e+00707KU-55933,LY294002,NU-7026,NU-7441,PI-103,PIK-75,PP-121,caffeine,compound-401,wortmannin
259Ube2hI3.996e-045940.000e+001819
260Ppp1caI3.970e-045690.000e+00913
261YwhaeI3.961e-046130.000e+001458
262Runx3I3.950e-042511.057e-0172
263PkmI3.935e-042011.331e-01665TEPP-46
264HnrnpuI3.920e-042131.452e-011028
265Lrrk2I3.915e-044990.000e+001860CZC-54252,GSK2578215A,LRRK2-IN-1,PF-06447475,URMC-099
266Cdh5I3.906e-048050.000e+00877fosbretabulin
267Cul1I3.889e-044560.000e+00849
268Birc3I3.869e-046440.000e+001244AZD5582,GDC-0152,SM-164
269Grb2I3.795e-048440.000e+001118
270TrrapI3.793e-047480.000e+00780
271NonoI3.786e-0410120.000e+00718
272Ddx39aI3.769e-041612.321e-011017
273Serbp1I3.758e-046590.000e+001392
274Myh9I3.708e-046270.000e+00811
275Nxf1I3.706e-043104.746e-021279
276Hnrnpa1I3.675e-048870.000e+001083
277Kmt5aI3.650e-043055.157e-0265
278Ect2I3.611e-044290.000e+00806
279YwhagI3.610e-048820.000e+001840
280Pik3r1I3.589e-046680.000e+00563CUDC-907,wortmannin
281Rac1I3.588e-043482.165e-021085EHop-016,dextromethorphan
282Ube2iI3.560e-047770.000e+00707
283Cbx2I3.500e-042826.594e-02125
284PcnaI3.489e-044880.000e+00786
285FlnaI3.480e-042777.107e-02730kartogenin
286Aurkaip1I3.472e-042241.050e-01287
287Cdk2I3.443e-042194.762e-02737AG-555,AT-7519,BMS-265246,BMS-387032,BMS-536924,BX-795,BX-912,CGP-60474,JNJ-7706621,NSC-625987
288Smad2I3.437e-044840.000e+00468dexfosfoserine
289Cdc123I3.428e-041502.878e-011701
290BsgI3.396e-042788.177e-02787
291Bap1I3.298e-044120.000e+001215
292Hspb1R3.296e-043163.991e-02867SB-242235,bicyclol
293Prc1I3.287e-046280.000e+00887PRT4165
294Xrcc6I3.273e-046840.000e+00982
295Nupr1I3.264e-041141.447e-01646
296Ddx6I3.258e-045930.000e+001437
297Egln3I3.249e-044490.000e+001254FG-4592
298Mov10I3.233e-048280.000e+001226
299MycnI3.223e-046020.000e+001289
300KrasI3.220e-042758.458e-021125K-Ras(G12C)-inhibitor-12,deltarasin,lonafarnib
301MtdhI3.195e-043462.338e-02506
302Afg2aI3.180e-049410.000e+001095
303FynI3.176e-046830.000e+00639bosutinib,dasatinib
304Mapk1I3.168e-048680.000e+007214,5,6,7-tetrabromobenzotriazole,BMS-536924,CHIR-99021,FR-180204,GDC-0994,KN-62,LY294002,PD-98059,SB-202190,SB-203580
305Fmr1I3.136e-043980.000e+00817
306Lgals1I3.111e-041202.302e-01390
307Sirt1I3.103e-047340.000e+00476EX-527,SRT1720,SRT2104,bisindolylmaleimide-IX,sirtinol,splitomycin,tenovin-1,tenovin-6
308Gsk3bI3.024e-045090.000e+008681-azakenpaullone,4,5,6,7-tetrabromobenzotriazole,7-hydroxystaurosporine,A-1070722,AR-A014418,AT7867,AZD1080,AZD2858,BX-795,BX-912
309Cdk1I3.022e-045520.000e+006041-azakenpaullone,7-hydroxystaurosporine,AT-7519,BMS-265246,CDK1-5-inhibitor,CGP-60474,CGP-74514,CHIR-99021,JNJ-7706621,P276-00
310SncaI3.021e-042905.435e-02840SMER-28
311H3c1I3.020e-048950.000e+001210
312Ruvbl1I3.014e-0410740.000e+00822
313Xrcc5I3.001e-049140.000e+00579
314Eef1a1I2.991e-042001.331e-01773
315Tuba1aI2.973e-049600.000e+00813albendazole,cabazitaxel,colchicine,docetaxel,mebendazole,paclitaxel,vinblastine,vinorelbine
316YwhahI2.963e-047060.000e+001395
317Ptpn11I2.939e-049560.000e+00614BVT-948,SHP099
318Huwe1I2.898e-041751.825e-011168
319HnrnpkI2.869e-046050.000e+00964
320Ybx1I2.829e-045100.000e+00785
321PmlI2.818e-0410430.000e+00893
322Csnk2a2I2.770e-042361.254e-01711CX-4945
323AlkI2.768e-04716.078e-01594AP26113,ASP3026,AZD3463,CEP-37440,GSK1838705A,KRCA-0008,NVP-TAE684,PF-06463922,adenosine-triphosphate,alectinib
324Tubb5I2.767e-047730.000e+008432-methoxyestradiol,ABT-751,CYT-997,D-64131,albendazole,cabazitaxel,carbendazim,cevipabulin,colchicine,docetaxel
325Rpl7aI2.755e-046900.000e+00700
326Snw1I2.753e-046630.000e+00905
327RictorI2.743e-044820.000e+00794
328AurkbI2.721e-048670.000e+00790AMG900,AT-9283,BI-847325,CCT129202,CCT137690,CGP-57380,CYC116,GSK1070916,GSK2334470,JNJ-7706621
329HadhaI2.714e-042679.312e-02636coenzyme-I
330Btf3I2.689e-048150.000e+00716
331Cops5I2.665e-044400.000e+001018
332Tnip1I2.656e-048550.000e+001073
333YwhaqI2.646e-047310.000e+001166
334Naa40I2.626e-049010.000e+00911
335Actc1I2.612e-047040.000e+00668
336Itm2bI2.611e-042737.743e-02886
337Phb1I2.605e-047720.000e+001161
338Cand1I2.591e-045240.000e+00877
339LynI2.580e-0410860.000e+00740bafetinib,bosutinib,dasatinib,ponatinib,rebastinib,tolimidone
340Trim21I2.578e-046740.000e+00634
341Fgfr1I2.570e-041529.317e-02623AZD4547,CH-5183284,LY2874455,MK-2461,NVP-BGJ398,PD-161570,PD-166285,PD-173074,RG1530,SUN-11602
342CyldI2.568e-047000.000e+00795
343Snai1I2.558e-047990.000e+00552
344Rpn1I2.557e-041821.134e-01862
345G3bp1I2.554e-049120.000e+00809
346YwhabI2.546e-047420.000e+001103
347EedI2.524e-041931.650e-011442EED226
348Ncor1I2.503e-048960.000e+00398
349CblI2.501e-049820.000e+00533
350Chmp4bI2.489e-043970.000e+00686
351Bag3I2.485e-044620.000e+00625
352Cav1I2.459e-043183.495e-02760
353Fbxo6I2.455e-041423.048e-01688
354Hnrnpa2b1I2.448e-049470.000e+00711
355Gja1I2.406e-046090.000e+008311-octanol,carbenoxolone,flufenamic-acid
356Notch1I2.396e-043303.020e-02366
357R3hdm2I2.394e-043373.404e-02116
358Usp48I2.385e-047450.000e+00684
359InsrI2.378e-049190.000e+00705GSK1838705A,GSK1904529A,NVP-AEW541,NVP-TAE684,ceritinib,dovitinib,linsitinib
360HadhbI2.363e-042797.071e-02544
361Hspa9I2.359e-041292.667e-01824
362HrasI2.358e-042728.955e-02994farnesyl-thiosalicylic-acid-amide,lonafarnib
363Bag6I2.348e-0410560.000e+00560
364Agr2I2.340e-048710.000e+00866
365Pcbp1I2.336e-048770.000e+00693
366Slc2a4I2.332e-047460.000e+005712-deoxyglucose
367Ruvbl2I2.330e-047820.000e+00804
368Rab11aI2.328e-042867.395e-02857
369Myef2I2.317e-043005.584e-0233
370Hdac4I2.305e-047560.000e+00745JNJ-26481585,LMK-235,SB-939,belinostat,dacinostat,givinostat,panobinostat,romidepsin,scriptaid,tasquinimod
371Rpn2I2.290e-042885.645e-02835
372Eftud2I2.290e-044630.000e+001495
373SfpqI2.259e-046860.000e+00532
374EmdI2.254e-044740.000e+00787
375NficI2.250e-046690.000e+00808
376Stip1I2.213e-046150.000e+001027
377Smarca2I2.204e-041014.521e-01392
378Hspd1I2.196e-043293.463e-021228
379OgtI2.191e-045300.000e+00941
380NfixI2.191e-049170.000e+00622
381H1-1I2.175e-04815.306e-01510
382Shank3I2.166e-049870.000e+00761
383Cbx3I2.161e-044260.000e+00621
384Wwp2I2.160e-043203.776e-02797
385Pik3caI2.155e-0411050.000e+00274A66,AS-604850,AZD6482,AZD8835,BGT226,CH5132799,ETP-45658,GDC-0349,GDC-0941,GDC-0980
386Rpl15I2.153e-045640.000e+00547anisomycin,puromycin
387Rpl13I2.149e-046330.000e+00767
388Stat1I2.148e-048120.000e+00435CKD-712
389Nr2c2I2.148e-043840.000e+001321retinol,tretinoin
390Ewsr1I2.124e-046190.000e+00842YK-4-279
391Map1bI2.111e-047260.000e+00555
392Epha2I2.105e-047150.000e+00711dasatinib,dorsomorphin,regorafenib,vandetanib
393SfnI2.100e-047870.000e+00807
394Rps13I2.091e-042321.394e-01736
395Actn4I2.088e-044060.000e+00422
396Smc1aI2.084e-044320.000e+00427
397Rnf2I2.081e-047800.000e+00836
398Prpf8I2.078e-046420.000e+00776
399Ubr4I2.075e-044860.000e+00335
400Rbm39I2.064e-044160.000e+00970
401BrafI2.062e-047940.000e+00529AZ-628,CEP-32496,GDC-0879,KG-5,LY3009120,ML786,PLX4720,PLX8394,RAF265,Ro-5126766
402H3-3aI2.057e-046950.000e+00949
403Ptpn1I2.056e-042624.230e-02647BVT-948,C11-Acetate,S-nitrosoglutathione,SNAP,bis(maltolato)oxovanadium(IV),corosolic-acid,evans-blue,hexylene-glycol,licochalcone-A,rheochrysidin
404FusI2.041e-049480.000e+00740
405CttnI2.040e-0410020.000e+00495
406Traf6I2.030e-044640.000e+00699
407Sumo2I2.024e-047700.000e+00585
408TardbpI2.015e-048340.000e+00676
409Gnb2I2.013e-042637.796e-02522
410Kpnb1I2.009e-048160.000e+00643
411Matr3I2.005e-045630.000e+00616
412Psmd1I2.002e-048190.000e+00478bortezomib
413TollipI1.999e-041661.399e-01435
414Mcm2I1.994e-044540.000e+00970
415PlecI1.988e-048400.000e+00481
416TmpoI1.980e-048080.000e+00754
417Psmd2I1.969e-046540.000e+00683bortezomib
418Disc1I1.965e-043213.261e-02822
419Iqgap1I1.964e-048880.000e+00633
420Psrc1I1.962e-043077.466e-0259
421Hoxa5I1.958e-043702.139e-02100
422RhobI1.955e-043681.039e-02825
423Rpl23I1.952e-042561.018e-01564anisomycin,puromycin
424MidnI1.951e-042161.460e-01569
425Kif20aI1.946e-043353.290e-02946
426SykI1.945e-045920.000e+003403,4-methylenedioxy-beta-nitrostyrene,BAY-61-3606,ER-27319,GDC-0980,GS-9973,PRT062070,PRT062607,R112,R406,ellagic-acid
427Hsph1I1.945e-046670.000e+00481
428Mib1I1.944e-042301.435e-01592
429Ppp1r9bI1.935e-048720.000e+00661
430Nup43I1.932e-047090.000e+00592
431Fxr1I1.929e-044140.000e+00742
432C9orf72I1.926e-044800.000e+001197
433PrkcaI1.919e-0410500.000e+004654,5,6,7-tetrabromobenzotriazole,7-hydroxystaurosporine,C-1,KN-62,LY294002,PD-98059,SB-202190,SB-203580,SC-10,SC-9
434Mki67I1.917e-049650.000e+00641
435SyncripI1.906e-045390.000e+00697
436AurkaI1.901e-046430.000e+00661AMG900,AT-9283,BI-847325,CCT129202,CCT137690,CYC116,ENMD-2076,GSK1070916,GSK2334470,JNJ-7706621
437JupI1.898e-048810.000e+00507
438Lamtor1I1.891e-042965.108e-02777
439Atg5I1.882e-042846.969e-02659
440Hmga2I1.880e-046400.000e+00582
441SbdsI1.877e-042184.762e-02951
442Pcbp4I1.869e-043542.898e-0241
443Rpl29I1.852e-043263.733e-0229
444Cul7I1.845e-041891.813e-01762
445Psma3I1.845e-044810.000e+00490bortezomib,carfilzomib
446Map3k7I1.841e-0411060.000e+00406RGB-286638
447Cacna1cR1.827e-042946.272e-02692BAY-K-8644-(s)-(-),FPL-64176,SNAP-5089,amlodipine,azelnidipine,benidipine,cleviprex,diltiazem,dronedarone,gabapentin
448H1-4I1.825e-041185.077e-01643
449Sirt6I1.811e-048370.000e+00594
450Nap1l1I1.810e-045780.000e+00373
451Hes6I1.807e-043551.912e-0250
452Nf2I1.806e-045570.000e+00450
453LrpprcI1.802e-046550.000e+00783
454Actg1I1.797e-0410830.000e+00567
455PpargI1.779e-049260.000e+00366BADGE,CINPA-1,FH-535,GW-1929,GW-9662,NPC-15199,S26948,SR-1664,T-0070907,acetyl-farnesyl-cysteine
456Pax6I1.773e-0410940.000e+00393
457Igf1rI1.764e-043014.127e-02436AG-1024,AZD3463,AZD4547,BMS-536924,BMS-754807,GSK1838705A,GSK1904529A,NT157,NVP-ADW742,NVP-AEW541
458CltcI1.750e-045450.000e+00729
459Ppp2r1aI1.743e-049430.000e+00642
460Arrb2I1.741e-048790.000e+00442
461Syngap1I1.740e-044100.000e+00668
462Dbn1I1.739e-049770.000e+00465
463Ddx21I1.729e-0410200.000e+001009
464IkbkgI1.717e-0410070.000e+00525flurizan
465Cct6aI1.710e-046660.000e+00569
466Sptan1I1.701e-047790.000e+00573
467Fbxo2I1.693e-04931.902e-01456
468Ptk2I1.685e-0410170.000e+00318ENMD-2076,NVP-TAE226,PF-431396,PF-562271,Y-11,defactinib
469Ranbp9I1.677e-04801.069e-01413
470Hsp90b1I1.668e-044890.000e+00728
471Lgals3bpI1.665e-044610.000e+00369
472Nr3c1I1.665e-049860.000e+0098817-hydroxyprogesterone-caproate,GSK9027,LXR-623,alclometasone-dipropionate,amcinonide,beclomethasone,beclomethasone-dipropionate,betamethasone,betamethasone-acetate,betamethasone-dipropionate
473Rpl28I1.658e-048470.000e+00528
474Pdia3I1.654e-0410700.000e+00490
475Bag1I1.637e-046880.000e+00447
476Hcn1I1.630e-042916.620e-02702ZD-7288,ivabradine,zatebradine
477Rpl8I1.628e-045030.000e+00574anisomycin,puromycin
478Rps15aI1.619e-044040.000e+00425
479DaxxI1.615e-045660.000e+00334
480HgsI1.608e-042812.449e-02526citric-acid
481Usp11I1.601e-049630.000e+00514
482Ube3aI1.597e-0410750.000e+00438
483Rps4xI1.590e-046960.000e+00570
484Usp9xI1.588e-0410030.000e+00442WP1130
485Psmc5I1.582e-046700.000e+00545
486Rab5aI1.580e-048750.000e+00712
487Zfpm2I1.574e-043591.278e-0237
488Frmd4aI1.573e-043711.958e-0227
489Dnmt1I1.573e-045560.000e+00280RG108,RX-3117,SGI-1027,azacitidine,decitabine,dimercaptosuccinic-acid,flucytosine,procainamide,triclabendazole,triclosan
490Fbxw11I1.566e-0410970.000e+00475
491HdlbpI1.564e-042094.898e-02827
492Tgfb1I1.562e-042576.984e-02304D-4476,F351
493Rbm14I1.557e-046870.000e+00580
494Rb1R1.556e-0410270.000e+00416
495Dctn1I1.554e-0410540.000e+00554
496RybpI1.543e-043313.020e-02643
497Runx2I1.543e-049880.000e+00219
498Tuba4aI1.543e-049640.000e+00558cabazitaxel,colchicine,docetaxel,paclitaxel,podophyllotoxin,vincristine,vinorelbine
499Msh2I1.540e-0410180.000e+00339
500NanogI1.539e-047550.000e+00315
501Rpl4I1.539e-047670.000e+00803
502Lamp2I1.539e-041034.054e-01802
503U2af2I1.538e-045250.000e+00783
504Csnk2bI1.538e-0410820.000e+00645
505Lima1I1.536e-044110.000e+00447
506Runx1I1.535e-046470.000e+00354
507Bag2I1.534e-047250.000e+00713
508Slc25a3I1.525e-048250.000e+00458
509Fbxl14I1.521e-043035.691e-0245
510Tgfbr2R1.508e-041282.582e-01366ITD-1,LY2109761
511Cbx1I1.506e-049310.000e+00401
512RhofI1.506e-0410900.000e+00652
513Eef1dI1.506e-046620.000e+00386
514Recql4I1.505e-045890.000e+001308
515Kpna1I1.504e-047680.000e+00395
516Lasp1I1.501e-048100.000e+00278
517Ddx39bI1.500e-048630.000e+00529
518Igf2bp3I1.495e-047810.000e+00504
519H1-2I1.495e-041761.949e-01624
520Cbx4I1.479e-049000.000e+00233
521Trim33I1.473e-049590.000e+00475
522Itgb1I1.469e-043392.174e-02451ATN-161,BIO-1211,BIO-5192,BTT-3033,SB-683698,TC-I-15,TCS-2314
523Igf2bp1I1.468e-045880.000e+00432
524CapzbI1.468e-046890.000e+001031
525Rplp0I1.466e-045170.000e+00823
526Eef1gI1.465e-043492.165e-02528
527Smarcb1I1.462e-047660.000e+00514
528UbbI1.461e-048560.000e+00903
529Mapk3I1.460e-046350.000e+00424CID-5458317,FR-180204,GDC-0994,arsenic-trioxide,purvalanol-B,ravoxertinib
530Mex3aI1.460e-049760.000e+00366
531Rpl6I1.457e-047490.000e+00673
532Arrb1I1.451e-043442.157e-02325
533Lmbr1lI1.448e-044900.000e+00919
534Cd81I1.446e-049670.000e+00468
535Rpl11I1.442e-048840.000e+00705anisomycin,puromycin
536NfiaI1.441e-044940.000e+00706
537Lmnb1I1.440e-0410490.000e+00611
538Hexim1I1.437e-047650.000e+00810
539Rpl3I1.436e-045680.000e+00743anisomycin,cycloheximide,homoharringtonine,puromycin
540Ddx5I1.426e-044010.000e+00637
541Ddb1I1.425e-044500.000e+00762
542Trap1I1.423e-0410530.000e+00493
543Pink1I1.423e-045160.000e+00596
544TnikI1.413e-044090.000e+00529
545Gcn1I1.410e-048970.000e+00456
546WwoxI1.406e-0410350.000e+00594
547Dhx15I1.400e-047370.000e+00552
548Cct4I1.399e-044530.000e+00649
549Hcfc1I1.396e-045530.000e+00330
550Lats2I1.395e-046260.000e+00291
551ZfxI1.391e-042876.162e-0217
552Phb2I1.390e-045810.000e+00640
553Fhl2I1.385e-044600.000e+00386
554Myo1bI1.384e-045540.000e+00295
555Cdk4I1.381e-0410110.000e+00295AMG-925,AT-7519,NSC-625987,ON123300,P276-00,PHA-793887,PHA-848125,R547,RGB-286638,SU9516
556Trim37I1.380e-045370.000e+00560
557Sf3b1I1.379e-042609.717e-02522
558Rbck1I1.370e-042895.435e-02515
559FblI1.362e-044050.000e+00630
560NacaI1.361e-049840.000e+00267
561Smarcd1I1.360e-049350.000e+00419
562Cct2I1.360e-044550.000e+00744
563Tle1I1.358e-0411310.000e+00223
564Twist2I1.352e-043834.712e-0329
565Polr2aI1.352e-047950.000e+00664dactinomycin
566MtorI1.350e-042657.143e-02369AP1903,AZ20,AZD2014,AZD8055,BGT226,CC-115,CC-223,CH5132799,GDC-0980,GSK2126458
567Slc25a5I1.349e-047740.000e+00526clodronic-acid
568Rps16I1.341e-047500.000e+00741
569Arf6I1.340e-046940.000e+00672
570Dhx9I1.335e-046300.000e+00701
571Cct3I1.329e-045750.000e+00758
572Tp53bp1I1.325e-048600.000e+00536
573ArntI1.323e-0410620.000e+00257
574Pabpc4I1.320e-046650.000e+00450
575Prmt1I1.319e-044970.000e+00866AMI-1,furamidine
576Gtf2bI1.316e-048260.000e+001082
577SprtnI1.315e-048480.000e+00538
578Wdr76I1.313e-042984.783e-02470
579Tnip2I1.308e-048040.000e+00870
580Sec61bI1.306e-043243.367e-02732
581Pdlim5I1.304e-0410460.000e+00293
582Ago2I1.302e-044410.000e+00539
583Sirt7I1.301e-047320.000e+00662
584TfrcI1.299e-048780.000e+00535
585Cul2I1.294e-046180.000e+00515
586Epas1I1.294e-045430.000e+00193PT-2385,TC-S-7009
587Psmd14I1.293e-047930.000e+00719
588DlstI1.291e-0410710.000e+00608
589Acta2R1.288e-0410800.000e+00339
590Foxp3I1.287e-049730.000e+00494
591Snrnp70I1.275e-043910.000e+00960
592Igf2bp2I1.275e-043144.205e-0212
593Rps20I1.272e-045060.000e+00778
594Il6raI1.271e-042317.273e-0230
595Rps14I1.269e-042281.382e-01578
596Myo1cI1.269e-047860.000e+00427
597GpkowI1.268e-049040.000e+00837
598Prpf19I1.267e-044200.000e+00508
599Numa1I1.266e-049100.000e+00479
600Myh10I1.264e-049240.000e+00408
601Rps6I1.261e-046310.000e+00897
602Fgf10I1.261e-043123.865e-0215
603HnrnpdlI1.260e-0410060.000e+00376
604Wfs1I1.259e-043511.834e-02517
605Dsg2I1.258e-0410340.000e+00293
606Cct5I1.257e-0410420.000e+00641
607Taf15I1.253e-044680.000e+00594
608Rps8I1.253e-046930.000e+00692
609Atp5f1cI1.249e-047140.000e+00532
610Znf800I1.248e-044270.000e+00338
611Mettl3I1.245e-04567.333e-01265
612Thrap3I1.239e-044930.000e+00469
613Caprin1I1.235e-043990.000e+00458
614ScribI1.234e-048570.000e+00593
615Cops6I1.233e-0410960.000e+00385
616Srsf1I1.226e-047440.000e+00771
617Mdn1I1.224e-045600.000e+00282
618Rab7aI1.221e-047690.000e+00922
619Gnb1I1.220e-043193.495e-02369
620Khdrbs1I1.215e-044150.000e+00417
621Tuba1bI1.214e-047620.000e+00518cabazitaxel,colchicine,docetaxel,paclitaxel,vinorelbine
622Tle3I1.205e-048530.000e+00365
623Atp1a1I1.205e-048540.000e+00613K-strophanthidin,almitrine,artemether,bretylium,chloroprocaine,ciclopirox,deslanoside,diazoxide,digitoxigenin,digitoxin
624QkiI1.203e-045610.000e+00657
625Smad1I1.202e-046070.000e+00273
626Larp1I1.201e-044250.000e+00474
627Dnm2I1.196e-0410810.000e+00410dynasore
628Tomm22I1.192e-043151.497e-02451
629Srsf3I1.192e-048290.000e+00541
630MepceI1.191e-044920.000e+00736
631Srsf7I1.186e-044030.000e+00884
632Hnf4aI1.186e-049280.000e+00317lauric-acid,linoleic-acid
633Rps19I1.183e-049080.000e+00670
634Zbtb7bI1.176e-049710.000e+00368
635Tubb4bI1.174e-044210.000e+00757albendazole,cabazitaxel,colchicine,docetaxel,mebendazole,oxibendazole,paclitaxel,vinorelbine
636ChukI1.170e-0410240.000e+00269BMS-345541,acetylcysteine,aminosalicylate,arctigenin,mesalazine,sulfasalazine
637Zdhhc5I1.168e-043432.462e-02558
638Prpf40aI1.167e-044830.000e+00527
639Vcam1I1.165e-047510.000e+00611succinobucol
640Ptges3I1.163e-0410580.000e+00454
641Hmga1I1.161e-044450.000e+00470
642Cse1lI1.155e-041512.727e-01359
643Tcf7l2I1.149e-047350.000e+00284
644Tp73I1.139e-049440.000e+00171
645Klf15I1.137e-049900.000e+00311
646Ilf2I1.131e-048060.000e+00610
647Gabarapl2I1.130e-046500.000e+00609
648CadI1.120e-048140.000e+00474L-aspartic-acid
649Men1I1.117e-049680.000e+00970
650Rpl30I1.117e-046910.000e+00568
651Wwtr1I1.116e-048350.000e+00434
652Nedd8I1.116e-044220.000e+00418
653Ddrgk1I1.115e-048460.000e+001160
654Rpl10aI1.110e-045400.000e+00528
655Cd44R1.108e-041917.715e-02294hyaluronic-acid
656Cdc73I1.106e-045440.000e+00439
657Tcp1I1.103e-046560.000e+00642
658Zc3h18I1.095e-047600.000e+00820
659Rpl12I1.092e-044910.000e+00453
660Rcor1I1.084e-048230.000e+00495
661NdnI1.084e-042926.620e-02437
662Heatr1I1.084e-0410790.000e+00415
663Hnrnpa0I1.082e-049330.000e+00305
664Ptbp1I1.082e-047640.000e+00398
665HnrnpfI1.078e-046760.000e+00573
666Eif4g1I1.075e-044470.000e+004544E1RCat
667Vdac1I1.073e-045460.000e+00572
668Ppp1cbI1.073e-0410510.000e+00516
669PrkacaI1.068e-049950.000e+00565A-674563,AT7867,CW-008,H-89,Y-27632,bucladesine,dexfosfoserine,ellagic-acid,fasudil,hydroxyfasudil
670Mcm3I1.067e-043890.000e+00423
671Rps15I1.061e-045120.000e+00682
672Rangap1I1.061e-049270.000e+00407
673HnrnpabI1.057e-047610.000e+00387
674Sf3b4I1.053e-046610.000e+00818
675PhgdhI1.051e-049970.000e+00412coenzyme-I
676Skp1I1.051e-044420.000e+00525
677Mcm5I1.050e-043900.000e+00453
678Rps23I1.047e-049790.000e+00409
679Dnajb1I1.046e-049990.000e+00349
680Slx4I1.046e-046320.000e+00627
681Nolc1I1.044e-046800.000e+00410
682Srpk1I1.044e-047750.000e+00479SRPIN340
683Eef2I1.041e-045380.000e+00661PJ-34
684Trim24I1.040e-048650.000e+00337
685Isg15I1.033e-047390.000e+00486
686Hyou1I1.029e-0410630.000e+00368
687Usp36I1.027e-045840.000e+00544
688Sin3aI1.027e-046450.000e+00396
689ErgI1.025e-046210.000e+00248
690Lrrc59I1.023e-049070.000e+00850
691Myo6I1.020e-045490.000e+00467
692Smndc1I1.019e-048410.000e+00769
693Bub3I1.019e-047240.000e+00267
694DspI1.019e-049200.000e+00469
695FasnI1.017e-046480.000e+004794-methylgenistein,GSK2194069,cerulenin,epicatechin-gallate-(-),epigallocatechin-gallate-(-),fisetin,morin,orlistat,pretomanid,pyrazinamide
696Plekha7I1.013e-048070.000e+00658
697Sptbn1I1.010e-047010.000e+00476
698Krt8I1.010e-049340.000e+00431
699HnrnprI1.008e-044440.000e+00476
700GsnR1.006e-043850.000e+00401
701Ranbp2I1.006e-049320.000e+00388
702Otub1I1.003e-049510.000e+00534
703Flot1I1.001e-041836.383e-02554
704Dkk1I9.915e-053534.237e-0221KY02111
705E2f1I9.884e-0511110.000e+00265
706Ctbp2I9.878e-056370.000e+00364
707Supt5hI9.872e-054350.000e+00485
708Sumo1I9.819e-058990.000e+00346
709E2f4I9.788e-058700.000e+00467
710Tfe3I9.786e-058320.000e+00382
711RbpjI9.782e-0510410.000e+00277
712Smarcd2I9.723e-0510680.000e+00196
713Copb1I9.684e-055280.000e+00410
714Rc3h1I9.680e-0510300.000e+00626
715Snrnp200I9.648e-0510450.000e+00506
716Vars1I9.630e-0510250.000e+00286
717Cfl1I9.567e-059400.000e+00399
718Usp10I9.557e-053452.157e-02296spautin-1
719Ipo5I9.528e-059940.000e+00441
720Asf1aI9.461e-0511200.000e+00278
721Rbx1I9.460e-054310.000e+00517
722Msh6I9.451e-055950.000e+00301
723Ube2oI9.450e-054240.000e+00739
724Banf1I9.435e-0510050.000e+00211
725Ufl1I9.411e-054510.000e+00959
726SafbI9.376e-059690.000e+00272
727Krt18I9.372e-059420.000e+00401
728HnrnpmI9.368e-056230.000e+00677
729Ksr1I9.342e-055140.000e+00462
730Rpl27aI9.341e-054080.000e+00529
731Gtf2iI9.319e-055340.000e+00419
732Tubb3I9.314e-059060.000e+00539cabazitaxel,colchicine,docetaxel,paclitaxel,vinorelbine
733Suz12I9.304e-056240.000e+00650
734Foxc1I9.288e-052159.292e-02240
735Rbbp4I9.282e-059150.000e+00576
736Srsf2I9.277e-055790.000e+00330
737Klf8I9.264e-052471.010e-01308
738Eif4bI9.205e-055150.000e+00415
739Foxa1I9.193e-057110.000e+00507
740Smurf1I9.142e-057410.000e+00535
741Ap2b1I9.113e-059460.000e+00429
742Nfe2l2I9.039e-052597.605e-02247NK-252,RTA-408,sulforaphane
743Usp15I8.996e-053920.000e+00526
744Wdtc1I8.937e-055270.000e+00560
745Pold1I8.923e-0510380.000e+00374clofarabine,cytarabine,fludarabine-phosphate
746Ccar2I8.888e-055740.000e+00375
747Ddx17I8.849e-057050.000e+00570
748Arid1aI8.835e-057900.000e+00256
749Ssrp1I8.820e-059030.000e+00666
750Hdac5I8.820e-054730.000e+00420JNJ-26481585,LMK-235,SB-939,belinostat,dacinostat,givinostat,romidepsin,scriptaid,trichostatin-a,vorinostat
751Upf1I8.814e-054070.000e+00637
752Actn1I8.706e-058730.000e+00385
753Fgfr3I8.633e-058660.000e+00575AEE788,AZD4547,CH-5183284,LY2874455,MK-2461,NVP-BGJ398,PD-173074,brivanib-alaninate,dovitinib,erdafitinib
754Rpl24I8.625e-052618.418e-02445
755Foxp1I8.599e-051472.740e-01249
756MecomI8.562e-056360.000e+00360
757Sugt1I8.515e-052229.630e-02391
758GanabI8.510e-0510840.000e+00391miglitol
759Ube2mI8.480e-0510770.000e+00601
760Slc3a2I8.477e-056290.000e+00440
761Aggf1I8.431e-059160.000e+00672
762Eprs1I8.420e-055290.000e+00522
763Nop56I8.371e-057970.000e+00613
764Pou5f1I8.364e-054180.000e+00352O4I1,OAC2
765Dpf2I8.361e-056160.000e+00337
766Tcf20I8.346e-053631.229e-0214
767Abce1I8.304e-054340.000e+00460
768H2axI8.292e-058240.000e+00640
769NrasI8.279e-052995.922e-02753lonafarnib
770Rps25I8.251e-058030.000e+00411
771Smc2I8.249e-055080.000e+00366
772Dync1h1I8.236e-054000.000e+00590
773Chaf1aI8.218e-058430.000e+00316
774Rcn1I8.130e-053114.508e-02267
775Usp14I8.070e-057160.000e+00482IU1,VLX600,WP1130
776Ppil4I8.061e-057920.000e+00763
777Hspa2I8.045e-058300.000e+00535
778Ccnd1I8.030e-058170.000e+00307arcyriaflavin-a,arsenic-trioxide,briciclib
779PrkraI7.984e-057880.000e+00372
780Abt1I7.981e-055820.000e+00456
781Sp7I7.964e-055620.000e+00310
782Rps5I7.964e-058010.000e+00514
783Chmp4cI7.958e-057910.000e+00598
784MetR7.903e-058980.000e+00432AMG-208,AMG-337,AMG458,BMS-536924,BMS-777607,BMS-817378,EMD-1214063,INC-280,JNJ-38877605,LY2801653
785CicI7.876e-054670.000e+00634
786Dot1lI7.836e-055770.000e+00755EPZ-5676,EPZ004777
787Srsf5I7.826e-059620.000e+00463
788Cdc37I7.824e-056410.000e+00673
789Srp14I7.816e-055000.000e+00350
790Rpl7I7.800e-059020.000e+00519
791Srrm2I7.772e-057220.000e+00480
792Sox4I7.730e-051442.703e-01178
793Sf3b2I7.724e-0510320.000e+00467
794BptfI7.680e-054960.000e+00215
795Mettl14I7.679e-056770.000e+00496
796Psmd4I7.674e-058000.000e+00474
797Zranb2I7.670e-057210.000e+00709
798Kcna3I7.628e-056220.000e+00843AS-77,CP-339818,dalfampridine
799Rps9I7.620e-058420.000e+00563
800Slc25a13I7.595e-0510570.000e+00319L-aspartic-acid
801Lonp1I7.587e-059180.000e+00507
802Smarcc1I7.562e-055860.000e+00392
803VdrR7.557e-0511280.000e+00150alfacalcidol,calcifediol,calcipotriol,calcitriol,cholecalciferol,dihydrotachysterol,doxercalciferol,eldecalcitol,ercalcitriol,ergocalciferol
804Hnrnpa3I7.551e-056990.000e+00463
805Cct8I7.522e-055320.000e+00748
806Yod1I7.513e-059090.000e+00477
807Rc3h2I7.497e-055200.000e+00615
808Atp5f1bI7.440e-058520.000e+00823
809Copb2I7.419e-0510210.000e+00505
810Phf21aI7.395e-0510230.000e+00349
811SrrtI7.390e-0510370.000e+00367
812HdgfI7.367e-052539.016e-02292
813Gpatch4I7.359e-059910.000e+00222
814Sec16aI7.355e-053860.000e+00459
815Psmc2I7.349e-055220.000e+00512
816Ncor2I7.327e-0510850.000e+00289
817Klf5I7.248e-057360.000e+00210
818Pcbp2I7.212e-055900.000e+00318
819Snrpd1I7.194e-0510360.000e+00387
820Cdk7I7.181e-058110.000e+00475BMS-387032,BS-181,PF-573228,PHA-793887,PHA-848125,R547,RGB-286638,TG-02,THZ1,THZ1-R
821ImmtI7.127e-056380.000e+00572
822Slc16a11I7.076e-055070.000e+00522
823Snrnp40I7.040e-056060.000e+00622
824Fubp3I7.011e-059960.000e+00307
825Smarca5I6.992e-054950.000e+00409
826Rpl13aI6.945e-058330.000e+00611anisomycin,puromycin
827Shmt2I6.887e-059550.000e+00660AZD4282,MC-1,mimosine
828Prrx1I6.858e-053255.676e-0225
829Rsl1d1I6.836e-055850.000e+00458
830Ssbp1I6.803e-055350.000e+00613
831Tra2aI6.800e-059210.000e+00442
832Dnaja1I6.797e-055230.000e+00568
833Sf3b3I6.765e-056570.000e+00527
834Eif3gI6.731e-058130.000e+00491
835Psmc6I6.718e-054520.000e+00405
836AatfI6.683e-055420.000e+00415
837Smc4I6.667e-055360.000e+00326
838Atp5poI6.649e-054650.000e+00444
839Atp5f1aI6.636e-055730.000e+00774
840Top2aI6.619e-056600.000e+00478aclarubicin,aldoxorubicin,amonafide,amrubicin,amsacrine,banoxantrone,ciprofloxacin,daunorubicin,dexrazoxane,doxorubicin
841Ncoa3I6.530e-056730.000e+00239
842Gata4I6.438e-056980.000e+00434
843Sf1I6.426e-059810.000e+00427
844CopaI6.422e-0510310.000e+00509
845Rbm15I6.344e-056460.000e+00695
846Eif2b4I6.304e-051791.818e-01164
847Akap8lI6.296e-0510090.000e+00289
848VapaI6.253e-059290.000e+00702
849TufmI6.208e-055580.000e+00742
850Ddx1I6.200e-058830.000e+00426
851Carm1I6.186e-059390.000e+00279sinefungin
852Dgcr8I6.186e-059250.000e+00702
853Rps18I6.180e-058510.000e+00440
854ZfrI6.170e-056030.000e+00275
855Brd3I6.139e-054170.000e+00445I-BET-762,I-BET151,LY303511,OTX015,XD-14,apabetalone
856Pik3r3I6.118e-051417.500e-02202
857Xrn2I6.082e-057200.000e+00421
858Nsun2I6.049e-055510.000e+00513
859Smarcc2I5.935e-059920.000e+00366
860Actl6aI5.928e-058930.000e+00281
861Rpl27I5.919e-055830.000e+00472
862Cct7I5.892e-055870.000e+00669
863Ddx18I5.885e-0510140.000e+00419
864Rps7I5.837e-059700.000e+00537
865Ccdc8I5.817e-059520.000e+00628
866Vps35I5.812e-057840.000e+00372
867Lin28aI5.747e-059530.000e+00696
868Uqcrc2I5.729e-056390.000e+00439
869Terf2ipI5.709e-054280.000e+00519
870Rad50I5.669e-055960.000e+00412
871Eif6I5.656e-054390.000e+00479
872Prdx1I5.648e-059360.000e+00401
873Csnk1a1I5.642e-057100.000e+00410D-4476,DRF053-(R),IC261
874Krr1I5.629e-059570.000e+00504
875Brd2I5.555e-054780.000e+00408I-BET-762,I-BET151,LY303511,OTX015,XD-14
876Smc5I5.548e-054190.000e+00908
877Rbbp5I5.539e-0510040.000e+00286
878H2az1I5.440e-056110.000e+00352
879RbmxI5.377e-054710.000e+00463
880Il12rb2I5.350e-053342.735e-0212
881SsbI5.340e-055720.000e+00505
882Cpsf6I5.238e-054720.000e+00578
883Iars1I5.200e-057290.000e+00414
884Bclaf1I5.185e-0510160.000e+00357
885Serpinh1I5.107e-057580.000e+00361
886Ddx27I5.073e-055010.000e+00374
887Exosc5I5.045e-055500.000e+00505
888Cbx5I5.026e-057170.000e+00343
889Slc16a1I5.024e-053273.644e-02233AR-C155858,AZD3965,CHC,UK-5099
890Ckap4I5.006e-058740.000e+00593
891TprI4.997e-0511090.000e+00314
892Adarb1I4.987e-054330.000e+00411
893Prkd1R4.981e-059890.000e+00188
894Igf2rI4.961e-051121.795e-01318
895Psma1I4.960e-058310.000e+00508bortezomib,carfilzomib
896FliiI4.943e-0510280.000e+00328
897Gnai3I4.929e-053362.688e-02277
898Kmt2aI4.905e-057890.000e+00320
899Hsf1I4.869e-055040.000e+00572
900Snd1I4.866e-053870.000e+00427
901Rad21I4.849e-057230.000e+00352
902H1-3I4.804e-054980.000e+00289
903Aar2I4.800e-059110.000e+00633
904Mta1I4.776e-0511000.000e+00294
905Rpl37aI4.758e-055050.000e+00373
906PpanI4.757e-058890.000e+00311
907Utp14aI4.737e-053561.503e-026
908AtmI4.711e-058640.000e+00345CGK-733,KU-55933,KU-60019,VE-822,caffeine
909Rrbp1I4.702e-058020.000e+00366
910AclyI4.693e-055470.000e+00397bempedoic-acid
911Hnrnpul1I4.642e-056780.000e+00373
912Prpf31I4.589e-0510640.000e+00380
913Srp72I4.587e-0510260.000e+00354
914AdarI4.578e-056200.000e+00304
915Ncbp1I4.575e-058910.000e+00538
916Uba1I4.554e-057780.000e+00453
917KhsrpI4.553e-0510470.000e+00325
918Mbd3I4.543e-057270.000e+00284
919Sart3I4.527e-059220.000e+00481
920Acin1I4.524e-054690.000e+00323
921Gnl3I4.521e-058850.000e+00591
922Dpp4I4.465e-052715.752e-024444-iodo-L-phenylalanine,DBPR108,NVP-DPP728,PK-44,UAMC-00039,alogliptin,anagliptin,atorvastatin,linagliptin,omarigliptin
923Aifm1I4.453e-056790.000e+00630flavin-adenine-dinucleotide
924Mybbp1aI4.434e-055410.000e+00477
925Ep400I4.412e-056750.000e+00208
926Fubp1I4.397e-0510330.000e+00311
927Rbm25I4.391e-054480.000e+00321
928DdostI4.378e-058380.000e+00474
929AsphI4.345e-056530.000e+00343L-aspartic-acid,succinic-acid
930Spp1R4.251e-056340.000e+00117
931Map4I4.219e-056810.000e+00366docetaxel,paclitaxel
932Noc2lI4.181e-055590.000e+00343
933PfkpI4.140e-056640.000e+00297
934Ehmt1I4.136e-059930.000e+00201A-366,BIX-01294,UNC0224,UNC0638,UNC0642,UNC0737
935Nufip2I4.102e-054770.000e+00356
936Eif2s1I4.081e-057130.000e+00349salubrinal
937Trim27I4.027e-056970.000e+00485
938Creb1I4.001e-058940.000e+00284adenosine-phosphate,naloxone
939Top1I3.972e-056100.000e+0066310-hydroxycamptothecin,9-aminocamptothecin,SN-38,TAS-103,aclarubicin,beta-lapachone,camptothecin,exatecan-mesylate,genz-644282,irinotecan
940Cul5I3.959e-056140.000e+00463
941Asxl1I3.912e-0510780.000e+00285
942Rpl22I3.716e-059230.000e+00452
943Rpl19I3.703e-057120.000e+00660anisomycin,puromycin
944Akap1I3.686e-055990.000e+00514
945Zc3hav1I3.681e-055190.000e+00596
946Prkaa2R3.647e-0511580.000e+00245aspirin
947Prmt5I3.463e-056250.000e+00496EPZ015666,HLCL-61
948Anxa2I3.443e-058220.000e+00441
949Tbx20I3.388e-0511449.287e-0330
950ShhI3.365e-053722.269e-0217SANT-1,SANT-2
951H2bc3I3.289e-058620.000e+00395
952Ccl2R3.200e-053521.522e-0259RS-504393,bindarit,danazol,mimosine
953Pate1I3.124e-052034.739e-02117
954Nop2I3.067e-055180.000e+00472
955GldcI3.061e-053223.553e-02317AZD4282,MC-1
956Srsf6I2.963e-059130.000e+00490
957Nat10I2.961e-054570.000e+00399remodelin
958Atad3aI2.939e-054380.000e+00533
959Kpna7I2.925e-053785.905e-038
960Srpk2I2.901e-057630.000e+00719SRPIN340,URMC-099,adenine,purvalanol-B
961Brms1I2.874e-053571.472e-0290
962Ncam1R2.871e-051261.538e-01134
963CoilI2.829e-057190.000e+00536
964Rpl36I2.799e-058500.000e+00477
965Lin28bI2.781e-058450.000e+00818
966Pes1I2.758e-055020.000e+00421
967Grwd1I2.697e-054750.000e+00430
968Macroh2a1I2.690e-0510100.000e+00413
969Pspc1I2.681e-055980.000e+00497
970Ddx54I2.632e-055650.000e+00570
971Smc3I2.624e-057540.000e+00403
972Nop58I2.605e-058800.000e+00411
973Pdcd11I2.553e-056170.000e+00439
974Eif4a1I2.544e-054370.000e+00403
975Dkc1I2.517e-057180.000e+00491
976Idh1R2.500e-056120.000e+00187AGI-5198,enasidenib,ivosidenib
977Rpl26I2.488e-057080.000e+00462anisomycin,puromycin
978Mad2l2I2.439e-052084.348e-02336
979Timp3R2.436e-0511080.000e+00103aminoguanidine
980LyarI2.401e-054130.000e+00428
981CtcfI2.391e-056720.000e+00430
982Mdc1I2.333e-0510190.000e+00427
983Ncoa1I2.313e-0510720.000e+00164T-0901317,corticosterone,genistein,indeglitazar,prinaberel
984Polr1gI2.263e-056710.000e+00463
985Itgb3R2.255e-0511240.000e+00193ATN-161,DU-728,GR-144053,cilengitide,eptifibatide,tirofiban
986Inf2R2.227e-055710.000e+00293
987Riok1I2.224e-057280.000e+00632
988Mre11I2.221e-055670.000e+00324
989Eif2ak2I2.201e-056920.000e+00288
990NifkI2.196e-056580.000e+00410
991MtrexI2.194e-057380.000e+00423
992Rrp12I2.129e-0510290.000e+00395
993Ddx56I2.108e-057830.000e+00360
994Eif2s2I2.100e-058200.000e+00334
995Srp68I2.079e-059580.000e+00429
996Sorl1I2.074e-053382.592e-02133
997Raver1I2.068e-059830.000e+00391
998Rbm28I2.045e-055210.000e+00368
999Rpl35aI2.026e-057400.000e+00442
1000Brix1I2.021e-055970.000e+00353
1001Ddx23I2.015e-056080.000e+00453
1002Eif3lI1.979e-054850.000e+00280
1003Slc27a2R1.969e-056000.000e+00283
1004Sipa1l2R1.960e-053422.429e-02139
1005Top2bI1.958e-054460.000e+00262amonafide,amrubicin,daunorubicin,dexrazoxane,etoposide,teniposide
1006Nudt21I1.933e-058920.000e+00335
1007Igfbp5R1.884e-0511460.000e+00133
1008Polr2bI1.882e-057300.000e+00442
1009AnpepI1.881e-05591.000e+00183ezetimibe,tosedostat
1010U2af1I1.876e-054660.000e+00372
1011Chn2I1.868e-053134.839e-0298
1012ApodR1.866e-0510910.000e+00168
1013Zbtb2I1.858e-059980.000e+00426
1014H1f10I1.858e-059300.000e+00286
1015Plxna1I1.856e-053411.869e-02130
1016Polr2cI1.839e-057030.000e+00533
1017Dnajc9I1.834e-058580.000e+00301
1018NesR1.823e-059780.000e+00165
1019Adamts1R1.810e-053621.087e-0293
1020Rbm4I1.791e-057020.000e+00294
1021Cbfa2t3R1.742e-0511630.000e+0086
1022Klf16I1.736e-0510890.000e+00401
1023NkrfI1.718e-057760.000e+00244
1024Polr1eI1.704e-056520.000e+00367
1025Zc3h14I1.689e-054590.000e+00795
1026Mfge8R1.684e-0511340.000e+0088
1027Ddx55I1.681e-054230.000e+00436
1028Gpc1R1.672e-059370.000e+00195
1029H3f4I1.669e-058210.000e+00402
1030Efnb2R1.659e-0511130.000e+00195
1031Suclg2I1.654e-051771.852e-01190succinic-acid
1032Mfap4I1.638e-051726.848e-02154
1033Hspa1lI1.601e-057520.000e+00342
1034Alx3I1.597e-053829.037e-0318
1035NischI1.576e-053737.605e-03190AGN-192403,agmatine,tizanidine
1036Fbxl6I1.552e-058900.000e+00551
1037AspmR1.520e-0510930.000e+00182
1038Tbl3I1.483e-056850.000e+00263
1039CenpfR1.431e-0511140.000e+00131
1040TfamI1.429e-055910.000e+00434
1041Nop53I1.416e-055700.000e+00359
1042Dkk3R1.366e-0510440.000e+0085
1043Plxna4R1.323e-053661.442e-0239
1044Dusp1R1.320e-0511540.000e+00101
1045Znf330I1.271e-059610.000e+00410
1046CenpaI1.265e-057530.000e+00347
1047Hipk2R1.260e-0510690.000e+0094
1048Aplp1I1.247e-053581.394e-0268
1049Rbm34I1.236e-059740.000e+00277
1050Fras1R1.199e-0511490.000e+0095
1051Itgb5R1.146e-0511300.000e+00133
1052Tead1I1.138e-059380.000e+00188
1053Hey1R1.109e-0511610.000e+00140
1054Nr4a1I1.093e-059750.000e+00232
1055AlcamR1.075e-0511720.000e+0080
1056Dnaja4R1.072e-058690.000e+0092
1057Atp6v1b1R1.048e-053479.950e-03132
1058Mageb4I1.039e-059660.000e+00363
1059Etv4I1.029e-0511520.000e+0084
1060Kgd4I1.008e-05798.333e-02132
1061Kcnj2R9.729e-0610080.000e+00242
1062Ptprz1R9.691e-067570.000e+0053
1063Ndc1I9.676e-063091.702e-02234
1064Samhd1R9.654e-065130.000e+00212
1065PtpruR9.334e-063746.349e-03125
1066GastI9.323e-063401.399e-0233acexamic-acid,sulmetozine
1067Col6a1R7.953e-0610390.000e+00124
1068KitR7.706e-0610870.000e+00126AC-710,APcK-110,CP-673451,DCC-2618,GTP-14564,KG-5,KI-20227,OSI-930,PLX647,amuvatinib
1069Arhgef6R7.591e-0611800.000e+00102
1070Igfbp4R7.533e-0611210.000e+0055
1071B4galt1I7.481e-06609.524e-0242N-acetyl-D-glucosamine
1072Prrx2R7.182e-0611850.000e+008
1073Sdc3R6.968e-067710.000e+0041
1074Frem2R6.872e-0611020.000e+0052
1075Klf12I6.831e-069720.000e+00202
1076Get3I6.451e-06571.000e+00152
1077Fbp2R5.699e-0611390.000e+0029
1078Vps26aI5.279e-063752.721e-03169
1079Man2a1I5.247e-063609.524e-03721-deoxymannojirimycin,kifunensine,swainsonine
1080Cyp24a1R5.197e-061782.778e-0263
1081Celsr1R5.184e-063619.524e-0367
1082Prom1R4.800e-0610950.000e+0041
1083Crip1R4.529e-0610010.000e+0051
1084Me1R4.366e-0611470.000e+0077coenzyme-I
1085Kiaa2013I4.317e-063674.975e-03146
1086Nqo1R4.256e-069450.000e+0090dicoumarol,flavin-adenine-dinucleotide,menadione
1087Unc5bR4.152e-0611620.000e+0095
1088Eme1I3.862e-063767.273e-0351
1089Emilin1R3.810e-063811.361e-03111
1090Cldn2R3.514e-063644.255e-0327
1091Gli2R3.506e-0611170.000e+00129GANT-61
1092Chi3l1R3.473e-0611260.000e+0034
1093Itga8R3.434e-063699.950e-0354
1094Ebf1I3.367e-06611.000e+0036
1095C1qtnf1R3.307e-063950.000e+0058
1096Pdzk1ip1R3.286e-0611730.000e+0086
1097Tnfrsf21R3.252e-0611320.000e+0030
1098Ube2uI3.149e-063501.639e-02110
1099Gpd1R2.857e-0610670.000e+0024coenzyme-I
1100PcolceR2.042e-063801.361e-0326
1101Ndufb8I2.025e-063795.155e-03138coenzyme-I
1102Plekhg1R1.873e-0610480.000e+0065
1103Atp6v1c2R1.813e-066820.000e+0041
1104Dnm1R1.803e-0610760.000e+00179dynasore,dynole-34-2,mdivi-1
1105Tfcp2l1R1.694e-0610660.000e+00105
1106Cd40R1.620e-065310.000e+00240
1107AldocR1.553e-069540.000e+00154
1108Mxra8R1.477e-063656.993e-0338
1109Fat4R1.455e-069850.000e+00101
1110VcanR1.316e-0610600.000e+0052hyaluronic-acid
1111Nt5eR1.298e-067850.000e+0090pentoxifylline
1112Prox1I1.127e-067980.000e+0060
1113VasnR7.944e-0710610.000e+00147
1114PxdnR7.829e-0711150.000e+0086
1115Fbn2R7.024e-0710590.000e+0077
1116Ankrd44R6.589e-078490.000e+0060
1117Sphk1R6.242e-0711380.000e+0089SKI-II,idronoxil
1118Foxi1R6.200e-0711480.000e+0089
1119Fads1R5.988e-0711330.000e+00108alpha-linolenic-acid,icosapent
1120Ntng1R4.454e-0710000.000e+00104
1121FibinR3.911e-0710980.000e+0064
1122Hsd17b7R2.953e-0711590.000e+0065coenzyme-I
1123Gramd1bR2.926e-0710990.000e+0092
1124PamR2.697e-0711680.000e+0059
1125LipaR2.554e-0710520.000e+0040
1126Kcnn4R2.530e-0711220.000e+00711-EBIO,AS-77,DCEBIO,NS-309,SKA-31,TRAM-34,TRAM-39,chlorzoxazone,clotrimazole,flindokalner
1127Celf2R2.425e-0710220.000e+0037
1128Ptgs1R2.368e-0711230.000e+0021O-acetyl-L-serine,SC-560,acemetacin,alclofenac,amfenac,aminosalicylate,ampiroxicam,amtolmetin-guacil,arachidonic-acid,aspirin
1129Pcdh18R2.346e-0711500.000e+0021
1130Cited2R2.187e-0711600.000e+0031
1131Garnl3R2.150e-075800.000e+0014
1132Mrc2R1.963e-0710130.000e+0065
1133Sema5aR1.957e-0711530.000e+0010
1134Susd5R1.953e-0711400.000e+0021
1135TgfbiR1.801e-0711010.000e+0024
1136Cyth3R1.629e-0711250.000e+0048
1137St3gal4R1.477e-0711430.000e+0051
1138Lhfpl2R1.407e-074700.000e+0036
1139Emp3R1.379e-0711030.000e+0068
1140Cxcl12R1.331e-0710550.000e+0029
1141Pdlim3R1.314e-0711290.000e+0025
1142Trpv4R1.220e-0711120.000e+003012-O-tetradecanoylphorbol-13-acetate,GSK2193874,HC-067047,RN-1734,RN-1747,capsazepine
1143Pdzd2R1.153e-0711870.000e+0023
1144Ckmt1R1.117e-0711100.000e+0019creatine
1145Vamp1R1.109e-0711760.000e+0059
1146Btn1a1R1.064e-0710150.000e+0023
1147PtgesR1.059e-0711820.000e+0020L-655240
1148Thbs2R9.999e-0811550.000e+0020
1149Lrg1R8.570e-0811270.000e+0012
1150Csmd1R8.130e-0811780.000e+008
1151Ttyh2R8.121e-0811670.000e+0022
1152Atp6v0a4R7.113e-0811180.000e+0032
1153Dlx3R7.081e-0811350.000e+0023
1154Vtcn1R6.362e-0811640.000e+0018
1155Slc25a36R5.503e-0811750.000e+007
1156Zcchc24R5.148e-0811420.000e+008
1157Ephx2R5.034e-0811980.000e+0023GSK2256294A
1158Rdh10R3.841e-085260.000e+0026
1159Ccdc3R3.402e-088360.000e+004
1160CckR2.902e-0811740.000e+0055
1161ChadR2.249e-0811190.000e+004
1162Heg1R2.112e-0811360.000e+0013
1163Sorcs2R1.715e-0811710.000e+0022
1164St8sia2R1.491e-0811410.000e+0010
1165B4galnt3R1.315e-0811940.000e+0018
1166Slc5a8R1.097e-0810880.000e+0047fenoprofen,ibuprofen-(S),ketoprofen
1167Them5R8.633e-0911450.000e+0019
1168Tpcn1R8.383e-0911070.000e+0034
1169Capn6R7.330e-0911040.000e+0026
1170Slc5a9R7.120e-0910650.000e+0028
1171Spock2R6.016e-0911830.000e+0020
1172Olfml3R5.737e-0910920.000e+0020
1173Abhd2R5.066e-0911690.000e+005
1174Rasgef1cR4.777e-0911840.000e+007
1175Atoh8R4.404e-0911790.000e+006
1176Clic6R3.516e-0911770.000e+0025
1177Osgin2R3.433e-0911860.000e+004
1178Egfl6R3.293e-0911510.000e+0019
1179Fut1R2.055e-0911570.000e+0031
1180Hepacam2R8.871e-1011660.000e+0036
1181GabrpR5.692e-1011880.000e+002acamprosate,amoxapine,butalbital,dehydroepiandrosterone,enflurane,etomidate,flumazenil,halothane,isoflurane,metharbital
1182Lrrc36R5.577e-1011920.000e+0010
1183Enpp3R4.474e-1011910.000e+008
1184Nudt4R3.298e-1011990.000e+003
1185Tll2R2.075e-1011700.000e+0019
1186Wdr72R1.953e-1010730.000e+008
1187Chrdl2R1.734e-1011810.000e+0035
1188Stard5R1.733e-1011370.000e+001
1189Pamr1R1.652e-1011160.000e+003
1190Muc15R1.629e-108270.000e+007
1191Tmem200bR4.203e-1111890.000e+003
1192FcgbpR4.229e-1211960.000e+001
1193LalbaR1.574e-1211560.000e+004
1194Wfdc3R1.259e-1211900.000e+001
1195Abcg2I0.000e+0011650.000e+001KS-176,cyclovalone
1196PtprvR0.000e+0011950.000e+000
1197TrfR0.000e+0011930.000e+000
1198Twist1D0.000e+005760.000e+00199
1199Wisp1R0.000e+0011970.000e+000
1200Zfp521R0.000e+0012000.000e+000

0.3 Assayed genes: every measurement (embedded)

Genelog2FCDrugIC50 (nM)Dissemination %NetPert rank
Sema5a2.77Gö-697611.480.01133
Ncam13.10SB-52533477.5113.6962
Emilin13.46Taxol6.01215.41089
Pcolce4.17Sorafenib151.226.71100
Ptprv2.53kb-NB142-70106.931.71196
Olfml33.44Genistein61433.31172
Fut14.34AMD31001628050.01179
Plekhg12.34C021.2HCl992.350.01102
Tgfbi2.73Batimastat176550.01135
Spock23.08Gö-6983104352.31171
Cbfa2t34.27CP 690550139759.11021
Mme3.19PF-5431082264.7149
Unc5b3.32SKI-5C19716570.01087
Plxna42.83GNF 58373108472.91043
Fat44.28CID-755636336981.21109
Cacna1c3.06CID-2011756978781.2447
Gramd1b2.76GM60013674983.31123
Col6a11.91Isradipine3280094.71067